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Epinastine HCl

CAS No. 108929-04-0

Epinastine HCl ( Epinastine Hydrochloride; Alesion; Elestat )

产品货号. M17804 CAS No. 108929-04-0

Epinastine is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.

纯度: 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
25MG ¥405 有现货
50MG ¥527 有现货
100MG ¥786 有现货
200MG ¥1482 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Epinastine HCl
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Epinastine is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
  • 产品描述
    Epinastine Hydrochloride is a histamine H1 receptor antagonist without sedative activity. Epinastine hydrochloride blocks the histamine H1 receptor and inhibits the release of histamine from mast cells. This prevents the typical allergic symptoms that are caused by histamine activity on capillaries, skin, and mucous membranes. Typical histamine activities include vasodilation, bronchoconstriction, increased vascular permeability, pain, itching, and spasmodic contractions of gastrointestinal smooth muscles. Epinastine HCl also has affinity for histamine H2, 5-HT2, and the alpha-1, alpha-2 adrenergic receptors.
  • 同义词
    Epinastine Hydrochloride; Alesion; Elestat
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    HT
  • 研究领域
    Inflammation/Immunology
  • 适应症
    ——

化学信息

  • CAS Number
    108929-04-0
  • 分子量
    285.77
  • 分子式
    C16H15N3·HCl
  • 纯度
    98%
  • 溶解度
    ——
  • SMILES
    Cl[H].NC1=NCC2N1C1=CC=CC=C1CC1=CC=CC=C21
  • 化学全称
    3-Amino-9,13b-dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepine Hydrochloride

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Fügner A, et al. Arzneimittelforschung, 1988, 38(10), 1446-1453.
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